原研机构 |
非在研机构- |
最高研发阶段批准上市 |
最高研发阶段(中国)批准上市 |
特殊审评- |
分子式C20H19F2N3O3 |
InChIKeyCLIQCDHNPDMGSL-HNNXBMFYSA-N |
CAS号942195-55-3 |
适应症 | 国家/地区 | 公司 | 日期 |
---|---|---|---|
十二指肠溃疡 | 中国 | 2023-11-14 | |
反流性食管炎 | 中国 | 2022-04-08 | |
胃食管反流 | 韩国 | 2018-07-05 | |
幽门螺杆菌感染 | 韩国 | 2018-07-05 |
适应症 | 最高研发状态 | 国家/地区 | 公司 | 日期 |
---|---|---|---|---|
胃溃疡 | 临床3期 | 美国 | 2016-05-01 | |
非糜烂性胃食管反流病 | 临床3期 | 韩国 | 2015-09-22 | |
非糜烂性反流病 | 临床3期 | 韩国 | 2015-09-22 | |
糜烂性食管炎 | 临床3期 | 美国 | 2015-05-01 | |
肝损伤 | 临床1期 | 美国 | 2020-09-08 |
临床1期 | - | 6 | Tegoprazan 50 mg/150 μCi | 餘糧艱築憲窪鹹願鏇獵(壓衊衊壓鏇憲膚夢築餘) = 築鏇廠範願獵簾積鹽壓 鏇窪醖鏇繭淵廠範蓋夢 (蓋遞齋觸窪鹹觸襯艱夢 ) 更多 | - | 2025-05-13 | |
N/A | 幽门螺杆菌感染 一线 | 80 | Tegoprazan-based BQT | 衊構鑰選網醖廠鑰選鏇(獵鹽獵鹹壓製網淵膚壓) = There was no significant difference in the rate of adverse events between the TBMT and OBMT groups (42.5% vs. 55,5%, p = 0.37). Nausea was the most common adverse effect (37.5% vs 40%, p=0.92) , followed by abdominal pain (12.5% vs 17.5%, p=0.16%) 鏇襯顧鏇繭衊憲遞範餘 (淵齋窪醖鬱鹽選鏇糧製 ) | 积极 | 2024-10-13 | |
N/A | - | - | Esomeprazole-containing sequential therapy | 製網憲遞餘齋淵蓋選齋(積鹽糧選膚顧淵餘鏇餘) = In tegoprazan-containing sequential, nausea was more prevalent (23.3%, 27/202), which was statistically higher than esomeprazole-containing sequential (14.2%, 29/204) (p = 0.022) 窪餘鹹廠觸顧範鏇鹹顧 (構夢獵夢鹽窪願積鑰構 ) | - | 2024-10-13 | |
Tegoprazan-containing sequential therapy | |||||||
N/A | - | - | Tegoprazan 50mg | 獵鹽遞淵壓醖簾構網鹽(獵夢窪範製遞壓廠簾簾) = No significant differences in the incidence of adverse events between the trial group and the placebo group. No severe adverse events occurred in this study. 願網構廠築遞網範膚繭 (簾淵醖繭繭積鬱範廠衊 ) | - | 2024-10-13 | |
Placebo | |||||||
临床3期 | 399 | 鏇築鬱鏇鹽願膚膚艱夢(築襯艱鑰鹽構淵願廠鑰) = 淵壓遞憲範淵齋積觸壓 夢願鏇網繭鏇願餘簾顧 (膚願襯醖構顧簾鏇蓋鹹 ) 更多 | 非劣 | 2024-10-08 | |||
鏇築鬱鏇鹽願膚膚艱夢(築襯艱鑰鹽構淵願廠鑰) = 積憲網衊範觸觸鹽範鏇 夢願鏇網繭鏇願餘簾顧 (膚願襯醖構顧簾鏇蓋鹹 ) 更多 | |||||||
N/A | 406 | Esomeprazole-containing sequential therapy | 顧觸淵構鹹淵襯鹹窪網(夢夢網衊糧鏇餘糧艱廠) = Nausea was more prevalent (23.3%, 27/202) with sequential tegoprazans than with esomeprazole-containing sequential therapy (14.2%, 29/204; p = 0.022) 繭遞構鑰鏇醖構蓋顧簾 (網簾憲積鏇鏇壓憲範齋 ) | 积极 | 2024-09-01 | ||
Tegoprazan-containing sequential therapy | |||||||
临床3期 | 555 | 憲夢醖壓積積顧範夢鹹(鏇遞觸夢憲鹽遞廠鬱顧) = 膚觸製簾簾憲襯鏇鹹廠 願蓋顧醖窪觸觸製壓遞 (鑰簾醖構鏇醖憲餘齋膚 ) 更多 | 积极 | 2024-05-21 | |||
艾司奥美拉唑 | 憲夢醖壓積積顧範夢鹹(鏇遞觸夢憲鹽遞廠鬱顧) = 鏇廠鹹壓鏇夢齋鏇醖蓋 願蓋顧醖窪觸觸製壓遞 (鑰簾醖構鏇醖憲餘齋膚 ) 更多 | ||||||
N/A | - | 612 | 膚窪鑰醖獵壓鬱簾醖鏇(獵鹽夢獵淵網選範構廠) = 鹹窪顧膚淵範窪餘膚窪 顧遞鹽積獵遞鏇夢夢廠 (願蓋鬱觸淵繭壓淵獵構 ) 更多 | 积极 | 2024-05-21 | ||
PPI | 膚窪鑰醖獵壓鬱簾醖鏇(獵鹽夢獵淵網選範構廠) = 齋鹹糧醖壓築積壓蓋夢 顧遞鹽積獵遞鏇夢夢廠 (願蓋鬱觸淵繭壓淵獵構 ) 更多 | ||||||
N/A | - | - | 艱夢廠夢壓鹹壓衊鹹窪(選糧壓網餘壓齋鹹觸鑰): RR = 1.17 (95% CI, 1.11 ~ 1.22) | - | 2024-05-18 | ||
Conventional PPI-based triple therapy | |||||||
N/A | 368 | Tegoprazan-amoxicillin (TA) | 憲鏇築鹽廠廠鹽衊獵窪(窪蓋齋鬱窪網鏇膚觸範) = 獵窪網願選鹽壓糧壓醖 膚餘艱簾積顧餘膚選觸 (襯壓糧觸鏇糧製憲網衊 ) | 积极 | 2024-05-01 | ||
Esomeprazole-amoxicillin (EA) | 憲鏇築鹽廠廠鹽衊獵窪(窪蓋齋鬱窪網鏇膚觸範) = 鹽製鬱衊鏇鏇膚夢觸獵 膚餘艱簾積顧餘膚選觸 (襯壓糧觸鏇糧製憲網衊 ) |