3区 · 化学
Article
作者: Chen, Kaixian ; Zheng, Mingyue ; Mao, Ruifeng ; Yang, Yaxi ; Luo, Xiaomin ; Ye, Yan ; Liu, Yu-Chih ; Xing, Jing ; Ding, Hong ; Wang, Yulan ; Jiang, Hualiang ; Zhang, Chenhua ; Zhou, Bing ; Luo, Cheng ; Zhang, Bidong
A series of highly selective and potent inhibitors against PRMT5 have been achieved using virtual screening and medicinal chemistry approaches.