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作者: Federico, Antonella ; Ducime, Alex ; Piccinini, Marco ; Pippione, Agnese C. ; Boschi, Donatella ; Al-Karadaghi, Salam ; Barge, Alessandro ; Sainas, Stefano ; Lolli, Marco L. ; Morice, Christophe ; Lupino, Elisa ; Contreras, Jean-Marie ; Kubbutat, Michael
Resulting from hit-to-lead optimization, the aminopyrazole3ais a NIK inhibitor selective over 44 kinases.